Sitagliptin-d4 phosphate 15528 BTCP binding was dose-dependently inhibited

BTCP binding was dose-dependently inhibited by unlabeled BTCP and nomifensine with the ID50 of 6

CAS Number: 1953-02-2

15(9): e0239147

BrH/c27-22(19-12-10-18(11-13-19)17-6-2-1-3-7-17)16-26-21-9-5-4-8-20(21)25-15-14-24-23(25)26

Sitagliptin-d4 phosphate 15528 BTCP binding was dose-dependently inhibitedSitagliptin d4 (MK 0431 d4) phosphate is the deuterium labeled Sitagliptin phosphate. Sitagliptin phosphate (MK 0431 phosphate) is a potent inhibitor of DPP4 with an IC50 of 19 nM in Caco 2 cell extracts. Product information CAS Number: 1432063 88 1 Molecular Weight: 508. 33 Formula: C16H17F6N5O5P Chemical Name: (3R) 3 amino 1 [3 (trifluoromethyl)(5,5,6,6 H) 5H,6H,7H,8H [1,2,4]triazolo[4,3 a]pyrazin 7 yl] 4 (2,4,5 trifluorophenyl)butan 1 one